Protein Details: Neuronal acetylcholine receptor subunit alpha-7

Protein ID

ICDB_Pro_0564

Protein Name

Neuronal acetylcholine receptor subunit alpha-7

Gene Name

Chrna7; Acra7

Organism

Mus musculus (Mouse)

Length

502 amino acids

AlphaFoldDB

AF-P49582-F1-model_v4.pdb

Function

Ionotropic receptor with a probable role in the modulation of auditory stimuli. Agonist binding induces a conformation change that leads to the opening of an ion-conducting channel across the plasma membrane. The channel is permeable to a range of divalent cations including calcium; the influx of which may activate a potassium current which hyperpolarizes the cell membrane. In the ear; this leads to a reduction in basilar membrane motion; altering the activity of auditory nerve fibers and reducing the range of dynamic hearing. This may protect against acoustic trauma. May also regulate keratinocyte adhesion. .

Sequence

MCGRRGGIWLALAAALLHVSLQGEFQRRLYKELVKNYNPLERPVANDSQPLTVYFSLSLLQIMDVDEKNQVLTTNIWLQMSWTDHYLQWNMSEYPGVKNVRFPDGQIWKPDILLYNSADERFDATFHTNVLVNASGHCQYLPPGIFKSSCYIDVRWFPFDVQQCKLKFGSWSYGGWSLDLQMQEADISSYIPNGEWDLMGIPGKRNEKFYECCKEPYPDVTYTVTMRRRTLYYGLNLLIPCVLISALALLVFLLPADSGEKISLGITVLLSLTVFMLLVAEIMPATSDSVPLIAQYFASTMIIVGLSVVVTVIVLRYHHHDPDGGKMPKWTRIILLNWCAWFLRMKRPGEDKVRPACQHKPRRCSLASVELSAGAGPPTSNGNLLYIGFRGLEGMHCAPTPDSGVVCGRLACSPTHDEHLMHGTHPSDGDPDLAKILEEVRYIANRFRCQDESEVICSEWKFAACVVDRLCLMAFSVFTIICTIGILMSAPNFVEAVSKDFA

PDB Structures

Ligand Binding

1. DICL_CP

2. DICL_Pep

Binding Site

SITE 86: "Key residue important for potent inhibition of the CHRNA9-CHRNA10 receptor by the alpha-conotoxin RgIA (AC P0C1D0)"; SITE 146: "Key residue important for potent inhibition of the CHRNA9-CHRNA10 receptor by the alpha-conotoxin RgIA (AC P0C1D0)"

Disease

Location

Detected in the nasal epithelium; in the outer hair cells of the cochlea; in the pars tuberalis of the hypophysis; and in the developing muscle of the tongue. Also expressed in the neurons of dorsal root ganglia.

DOI ID

10.1016/0092-8674(94)90555-x; 10.1016/s0378-5955(99)00214-2; 10.1016/s0028-3908(00)00124-6; 10.1073/pnas.051622798; 10.1016/s0378-5955(02)00380-5; 10.1016/s0306-4522(02)00274-9; 10.1124/mol.65.2.453; 10.1111/j.1471-4159.2012.07867.x; 10.1016/j.jmb.2008.01.082; 10.1124/mol.114.096511; 10.1124/mol.114.096511err

RefSeq

NP_075219.1

Feature